PTCE Top 200 · #191

Nebivolol

Bystolic

Nebivolol is the generic name for the brand-name drug Bystolic. It is a beta blocker (beta-1 selective) used to treat hypertension. On the PTCE Top 200 drug list, Nebivolol ranks #191 and is one of the most frequently tested cardiovascular medications — commonly quizzed on its brand–generic pair, drug class, and key side effects.

Generic nameNebivolol
Brand name(s)Bystolic
Drug classBeta blocker (beta-1 selective)
Class groupCardiovascular
Common usehypertension
DEA scheduleUnscheduled
AvailabilityPrescription only (Rx)

What is Nebivolol used for?

Treatment of hypertension (the US-approved indication). Heart-failure use is off-label / outside the US.

What drug class is Nebivolol?

Nebivolol is a Beta blocker (beta-1 selective) in the Cardiovascular group. Knowing the class is the fastest way to predict its uses, side effects, and the brand↔generic pairs the PTCE tests.

Common side effects of Nebivolol

Major interactions

Is Nebivolol a controlled substance?

No. Nebivolol is not a federally controlled substance (it is unscheduled by the DEA).

How to remember Nebivolol (PTCE mnemonic)

BY-stolic BYpasses sympathetic surge — NEBIvolol is β1-selective + NO-mediated vasodilation (unique). Less fatigue/ED than other β-blockers; slows HR; never stop abruptly.
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PTCE exam tip

Nebivolol is the 'gentle' cardioselective beta blocker with added vasodilation — it still ends in -olol, and like the class it's tapered, never stopped abruptly.

Nebivolol FAQ

What is the brand name for Nebivolol?

The brand name for Nebivolol is Bystolic.

What is Nebivolol used for?

Nebivolol is used to treat hypertension. Treatment of hypertension (the US-approved indication). Heart-failure use is off-label / outside the US.

What drug class is Nebivolol?

Nebivolol is a Beta blocker (beta-1 selective) (Cardiovascular group).

Is Nebivolol a controlled substance?

No. Nebivolol is not a federally controlled substance (it is unscheduled by the DEA).

Related drugs in the Cardiovascular group

Drill Nebivolol the way the PTCE asks it

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Last reviewed June 25, 2026. Educational use only — not medical advice. Verify clinical specifics with your pharmacist or a current label source such as DailyMed. RxReflex is not affiliated with or endorsed by the Pharmacy Technician Certification Board (PTCB).